Systems-pharmacology dissection of a drug synergy in imatinib-resistant CML
Scansite Kinase
| Domain | Peptides | |
|---|---|---|
| None | 342 | |
| Casn_Kin2 | 63 | |
| Cdc2_Kin | 44 | |
| Erk1_Kin | 42 | |
| Cdk5_Kin | 41 | |
| Akt_Kin | 31 | |
| PKA_Kin | 25 | |
| AMPK | 20 | |
| GSK3_Kin | 18 | |
| Clk2_Kin | 17 | |
| Cam_Kin2 | 8 | |
| p38_Kin | 6 | |
| Lck_Kin | 4 | |
| Src_Kin | 4 | |
| Casn_Kin1 | 3 | |
| Abl_Kin | 3 | |
| ATM_Kin | 3 | |
| Itk_Kin | 1 | |
| InsR_Kin | 1 |
Scansite Bind
| Domain | Peptides | |
|---|---|---|
| None | 431 | |
| CDK1_1 | 48 | |
| CDK1_2 | 42 | |
| AuroA | 21 | |
| 1433_m1 | 21 | |
| GSK3b | 18 | |
| AuroB | 15 | |
| DNA_PK | 13 | |
| PKC_epsilon | 3 | |
| Fgr_SH2 | 2 | |
| Fyn_SH2 | 2 | |
| PLCg_NSH2 | 1 | |
| Grb2_SH2 | 1 | |
| Abl_SH2 | 1 | |
| Crk_SH2 | 1 | |
| Nck_SH2 | 1 | |
| Lck_SH2 | 1 | |
| p85_SH2 | 1 | |
| Shc_SH2 | 1 | |
| PKC_delta | 1 | |
| PDK1_Bind | 1 |